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Trypsin inhibitors:
PDB ID: 1C2D Citation: Katz, B.A., Luong, C. Recruiting Zinc to Mediate Potent, Specific Inhibition of Serine Proteases (1999) doi 10.2210/pdb1C2D/pdb
PDB ID: 1C5T Citation: Katz, B.A., Mackman, R., Luong, C., Radika, K., Martelli, A., Sprengeler, P.A., Wang, J., Chan, H., Wong, L. Structural Basis for Selectivity of a Small Molecule, S1-Binding, Sub-Micromolar Inhibitor of Urokinase Type Plasminogen Activator (1999) doi 10.2210/pdb1C5T/pdb
PDB ID: 1F0T Citation: Maignan, S., Guilloteau, J.P., Pouzieux, S., Choi-Sledeski, Y.M., Becker, M.R., Klein, S.I., Ewing, W.R., Pauls, H.W., Spada, A.P., Mikol, V. Bovine Trypsin Complexed with RPR131247 (2000) doi 10.2210/pdb1F0T/pdb
PDB ID: 1G3D Citation: Toyota, E., Ng, K.K.S., Sekizaki, H., Itoh, K., Tanizawa, K., James, M.N.G. Bovine Beta-Trypsin Bound to Meta-Amidino Schiff Base Copper (II) Chelate (2000) doi 10.2210/pdb1G3D/pdb
PDB ID: 1G3E Citation: Toyota, E., Ng, K.K.S., Sekizaki, H., Itoh, K., Tanizawa, K., James, M.N.G. Bovine Beta-Trypsin Bound to Para-Amidino Schiff Base Copper (II) Chelate (2000) doi 10.2210/pdb1G3E/pdb
PDB ID: 1GHZ Citation: Katz, B.A., Elrod, K., Luong, C., Rice, M., Mackman, R.L., Sprengeler, P.A., Spencer, J., Hatayte, J., Janc, J., Link, J., Litvak, J., Rai, R., Rice, K., Sideris, S., Verner, E., Young, W. A Novel Serine Protease Inhibition Motif Involving a Multi-Centered Short Hydrogen Bonding Network at the Active Site (2001) doi 10.2210/pdb1GHZ/pdb
PDB ID: 1GJ6 Citation: Katz, B.A., Sprengeler, P.A., Luong, C., Verner, E., Spencer, J.R., Breitenbucher, J.G., Hui, H., McGee, D., Allen, D., Martelli, A., Mackman, R.L. Engineering Inhibitors Highly Selective for the S1 Sites of SER190 Trypsin-Like Serine Protease Drug Targets (2001) doi 10.2210/pdb1GJ6/pdb
PDB ID: 1H4W Citation: Katona, G., Berglund, G.I., Hajdu, J., Graf, L., Szilagyi, L. Structure of human trypsin IV (brain trypsin) (2001) doi 10.2210/pdb1H4W/pdb
PDB ID: 1J17 Citation: Stubbs, M.T. Factor XA Specific Inhibitor in Complex with Rat Trypsin Mutant X99/175/190RT (2002) doi 10.2210/pdb1J17/pdb
PDB ID: 1K1I Citation: Stubbs, M.T. Bovine Trypsin-Inhibitor Complex (2001) doi 10.2210/pdb1K1I/pdb
PDB ID: 1K1L Citation: Stubbs, M.T. Bovine Trypsin-Inhibitor Complex (2001) doi 10.2210/pdb1K1L/pdb
PDB ID: 1K1N Citation: Stubbs, M.T. Bovine Trypsin-Inhibitor Complex (2001) doi 10.2210/pdb1K1N/pdb
PDB ID: 1PPC Citation: Bode, W., Turk, D. Geometry of Binding of the Benzamidine-and Arginine-Based Inhibitors N-alpha-(2-naphthyl-sulphonyl-glycyl)-DL-P-amidinophenylalanyl-oiperidine (NAPAP) and (2R,4R)-4-methy-1-[N-alpha-(3-methyl-1,2,3,4-tetrahydro-8-quinolinesulphonyl)-L-arginyl]-2-piperidine Carboxylic Acid (MQPA) to Human Alpha-Thrombin: X-Ray Crystallographic Determination of the NAPAP-Trypsin Complex and Modeling of NAPAP-Thrombin AND MQPA-Thrombin (1991) doi 10.2210/pdb1PPC/pdb
PDB ID: 1QB1 Citation: Whitlow, M. Bovine Trypsin with 1-[2-[5-[amino(imino)methyl]-2-hydroxyphenoxy]-6-[3-(4,5-dihydro-1-methyl-1H-imidazol-2-yl)phenoxy]pyridin-4-yl]piperidine-3-carboxylic Acid (ZK-806974) (1999) doi 10.2210/pdb1QB1/pdb
PDB ID: 1QB6 Citation: Whitlow, M. Bovine Trypsin 3,3’-[3,5-difluoro-4-methyl-2, 6-pyridinediylbis(oxy)]bis(benzenecarboximidamide) (ZK-805623) Complex (1999) doi 10.2210/pdb1QB6/pdb
PDB ID: 1QB9 Citation: Whitlow, M. Bovine Trypsin 7-[[2-[[1-(1-iminoethyl)piperidin-4-YL]oxy]-9H-carbozol-9-YL] methyl]naphthalene-2-carboximidamid (ZK-806450) Complex (1999) doi 10.2210/pdb1QB9/pdb
PDB ID: 1QBN Citation: Whitlow, M. Bovine Trypsin 2-[amino(imino)methyl]-2-hydroxyphenoxy]-6-[3-(4,5-dihydro-1H-imidazol-2-yl)phenoxy]pyridine-4-carboxylic Acid (ZK-806688) Complex (1999) doi 10.2210/pdb1QBN/pdb
PDB ID: 1QBO Citation: Whitlow, M. Bovine Trypsin 7-[[6-[[1-(1-iminoethyl)piperidin-4-YL]oxy]-2-methyl-benzimidazol-1-YL]methyl]naphthalene-2-carboximidamid ZK-806711 Inhibitor Complex (1999) doi 10.2210/pdb1QBO/pdb
PDB ID: 1TNI Citation: Kurinov, I., Harrison, R.W. Prediction of Novel Serine Protease Inhibitors (1994) doi 10.2210/pdb1TNI/pdb
Estrogen antagonist receptor:
PDB ID: 3ERT Citation: Shiau, A.K., Barstad, D., Loria, P.M., Cheng, L., Kushner, P.J., Agard, D.A., Greene, G.L. Human Estrogen Receptor Alpha Ligand-Binding Domain in Complex with 4-Hydroxytamoxifen. (1999) doi 10.2210/pdb3ERT/pdb
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